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Atomfair Revefenacin TD-4208, GSK-1160724 C35H43N5O4 CAS 864750-70-9

Revefenacin (CAS No. 864750-70-9) is a long-acting muscarinic antagonist (LAMA) with the molecular formula C35H43N5O4and the IUPAC name [1-[2-[[4-[(4-carbamoylpiperidin-1-yl)methyl]benzoyl]-methylamino]ethyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate. This high-purity compound is specifically designed for research and pharmaceutical development, offering exceptional selectivity and potency in targeting muscarinic receptors. Revefenacin is supplied as a fine powder with guaranteed ≥98% purity (HPLC), ensuring reliability for in vitro and in vivo studies. Its low water solubility makes it ideal for formulation in organic solvents such as DMSO or ethanol. Suitable for COPD research, receptor binding assays, and pharmacokinetic studies, this product is rigorously tested for stability, endotoxin levels, and residual solvents…

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Description

Revefenacin (CAS No. 864750-70-9) is a long-acting muscarinic antagonist (LAMA) with the molecular formula C35H43N5O4 and the IUPAC name [1-[2-[[4-[(4-carbamoylpiperidin-1-yl)methyl]benzoyl]-methylamino]ethyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate. This high-purity compound is specifically designed for research and pharmaceutical development, offering exceptional selectivity and potency in targeting muscarinic receptors. Revefenacin is supplied as a fine powder with guaranteed ≥98% purity (HPLC), ensuring reliability for in vitro and in vivo studies. Its low water solubility makes it ideal for formulation in organic solvents such as DMSO or ethanol. Suitable for COPD research, receptor binding assays, and pharmacokinetic studies, this product is rigorously tested for stability, endotoxin levels, and residual solvents to meet the highest industry standards.

Properties

  • CAS Number: 864750-70-9
  • Complexity: 918
  • IUPAC Name: [1-[2-[[4-[(4-carbamoyl-1-piperidyl)methyl]benzoyl]-methyl-amino]ethyl]-4-piperidyl] N-(2-phenylphenyl)carbamate
  • InChI: InChI=1S/C35H43N5O4/c1-38(34(42)29-13-11-26(12-14-29)25-40-19-15-28(16-20-40)33(36)41)23-24-39-21-17-30(18-22-39)44-35(43)37-32-10-6-5-9-31(32)27-7-3-2-4-8-27/h2-14,28,30H,15-25H2,1H3,(H2,36,41)(H,37,43)
  • InChI Key: FYDWDCIFZSGNBU-UHFFFAOYSA-N
  • Exact Mass: 597.33150487
  • Molecular Formula: C35H43N5O4
  • Molecular Weight: 597.7
  • SMILES: CN(CCN1CCC(CC1)OC(=O)NC2=CC=CC=C2C3=CC=CC=C3)C(=O)C4=CC=C(C=C4)CN5CCC(CC5)C(=O)N
  • Topological: 108
  • Monoisotopic Mass: 597.33150487
  • Solubility: < 1 mg/ml
  • Synonyms: Revefenacin, TD-4208, Yupelri, GSK-1160724, revefenacina, revefenacine, GSK1160724, G2AE2VE07O, UNII-G2AE2VE07O, 1-(2-(4-((4-Carbamoylpiperidin-1-yl)methyl)-N-methylbenzamido)ethyl)piperidin-4-yl N-((1,1′-biphenyl)-2-yl)carbamate, TD4208, Biphenyl-2-ylcarbamic acid 1-(2-((4-(4-carbamoylpiperidin-1-ylmethyl)benzoyl)methylamino)ethyl)piperidin-4-yl ester, Biphenyl-2-ylcarbamic acid, 1-(2-((4-(4-carbamoylpiperidin-1-ylmethyl)benzoyl)methylamino)ethyl)piperidin-4-yl ester, Carbamic acid, N-(1,1′-biphenyl)-2-yl-, 1-(2-((4-((4-(aminocarbonyl)-1-piperidinyl)methyl)benzoyl)methylamino)ethyl)-4-piperidinyl ester, revefenacinum, R03BB08, 864750-70-9, Revefenacin [INN], 1-(2-(3-((4-carbamoylpiperidin-1-yl)methyl)-N-methylbenzamido)ethyl)piperidin-4-yl [1,1′-biphenyl]-2-ylcarbamate, Revefenacin [WHO-DD], 864750-70-9 (free base), [1-[2-[[4-[(4-carbamoylpiperidin-1-yl)methyl]benzoyl]-methylamino]ethyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate, 1-(2-(4-((4-Carbamoylpiperidin-1-yl)methyl)-N-methylbenzamido)ethyl)piperidin-4-yl [1,1′-biphenyl]-2-ylcarbamate, TD-4208; GSK-1160724;[1-[2-[[4-[(4-carbamoylpiperidin-1-yl)methyl]benzoyl]-methylamino]ethyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate, Carbamic acid, N-[1,1′-biphenyl]-2-yl-, 1-[2-[[4-[[4-(aminocarbonyl)-1-piperidinyl]methyl]benzoyl]methylamino]ethyl]-4-piperidinyl ester; Carbamic acid, [1,1′-biphenyl]-2-yl-, 1-[2-[[4-[[4-(aminocarbonyl)-1-piperidinyl]methyl]benzoyl]methylamino]ethyl]-4-, Yupelri (TN), Revefenacin (Standard), REVEFENACIN [MI], Revefenacin (USAN/INN), Revefenacin [USAN:INN], REVEFENACIN [USAN], Revefenacin;GSK1160724, SCHEMBL356480, CHEMBL3833319, GTPL10129, REVEFENACIN [ORANGE BOOK], DTXSID701027775, GLXC-23321, HMS3886K17, HMS5084F21, Revefenacin [USAN:INN:WHO-DD], BCP15793, EX-A1722, HY-15851R, s5258, AKOS037649398, CCG-270187, CS-7743, DB11855, SB17262, BS-18189, DA-57407, FR178690, HY-15851, TD-4208?, NS00073361, D10978, EN300-20352165, Q27278649, Revefenacin; TD 4208; TD4208; GSK-1160724; GSK1160724; GSK 1160724, 1-[2-(1-{4-[(4-carbamoylpiperidin-1-yl)methyl]phenyl}-N-methylformamido)ethyl]piperidin-4-yl N-{[1,1′-biphenyl]-2-yl}carbamate, 1211931-83-7, TD-4208;1-(2-(3-((4-carbamoylpiperidin-1-yl)methyl)-N-methylbenzamido)ethyl)piperidin-4-yl [1,1-biphenyl]-2-ylcarbamate

Application

Revefenacin is primarily used as a long-acting muscarinic antagonist (LAMA) for the treatment of chronic obstructive pulmonary disease (COPD). It functions by inhibiting bronchoconstriction, thereby improving lung function and reducing symptoms. Researchers utilize Revefenacin in preclinical and clinical studies to investigate its efficacy and safety profile. It is also employed in receptor binding assays to study muscarinic receptor interactions and signaling pathways.

Safety and Hazards

GHS Hazard Statements

  • H302 (100%): Harmful if swallowed [Warning Acute toxicity, oral]
  • H312 (100%): Harmful in contact with skin [Warning Acute toxicity, dermal]
  • H332 (100%): Harmful if inhaled [Warning Acute toxicity, inhalation]

Precautionary Statements

  • P261, P264, P270, P271, P280, P301+P317, P302+P352, P304+P340, P317, P321, P330, P362+P364, and P501

Hazard Classes and Categories

  • Acute Tox. 4 (100%)

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Disclaimer: Sold exclusively for laboratory research. Prohibited for commercial use, diagnostics, or human/animal applications. Buyers assume all compliance liability.

Disclaimer

Intended Use & Restrictions

This product is sold exclusively for laboratory research, analytical testing, or non-commercial purposes.

  • Strictly prohibited: Resale, repackaging, or formulation into commercial products.
  • Not approved for human/animal use, diagnostics, or manufacturing (including pharmaceuticals, agrochemicals, or consumer goods).

Patent & Regulatory Compliance

Certain molecules may be protected by active patents or regulatory restrictions.

  • Buyers must independently verify patent status (e.g., via USPTO/EPO/CNIPA) and comply with local laws.
  • Atomfair LLC does not provide legal assurances regarding patent non-infringement or jurisdictional compliance.

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  • Use this product only as permitted by law.
  • Indemnify Atomfair LLC against all claims arising from misuse, patent infringement, or regulatory violations.

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